Search Result "biased agonism"


A Pharmacological Primer of Biased Agonism

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 11 Issue: 2 Year: 2011 Page: 92-98
Author(s): Bradley T. Andresen

Biased Agonism of the Angiotensin II Type 1 Receptor

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 9 Year: 2012 Page: 812-816
Author(s): C. M. Godin,S. S.G. Ferguson

Review Article

Biased Agonism as an Emerging Strategy in the Search for Better Opioid Analgesics

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 9 Year: 2020 Page: 1562-1575
Author(s): Justyna Piekielna-Ciesielska,Karol Wtorek,Anna Janecka

Novel Insights into Biased Agonism at G Protein-Coupled Receptors and their Potential for Drug Design

Journal: Current Pharmaceutical Design
Volume: 19 Issue: 2 Year: 2013 Page: 5156-5166
Author(s): Maria Marti-Solano, Ramon Guixa-Gonzalez, Ferran Sanz, Manuel Pastor, Jana Selent

Biased Agonism at the Parathyroid Hormone Receptor: A Demonstration of Functional Selectivity in Bone Metabolism

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 9 Year: 2012 Page: 856-865
Author(s): B. N. Bohinc,D. Gesty-Palmer

Beta-arrestin Biased Agonism/Antagonism at Cardiovascular Seven Transmembrane-spanning Receptors

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 2 Year: 2012 Page: 192-198
Author(s): Anastasios Lymperopoulos

Review Article

Innovative Opioid Peptides and Biased Agonism: Novel Avenues for More Effective and Safer Analgesics to Treat Chronic Pain

Journal: Current Medicinal Chemistry
Volume: 25 Issue: 3 Year: 2018 Page: 3895-3916
Author(s): Andrea Bedini,Santi Spampinato

β-arrestin-Biased Agonism at the Parathyroid Hormone Receptor Uncouples Bone Formation from Bone Resorption

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 11 Issue: 2 Year: 2011 Page: 112-119
Author(s): Brittany N. Bohinc, Diane Gesty-Palmer

Review Article

From Receptor Selectivity to Functional Selectivity: The Rise of Biased Agonism in 5-HT1A Receptor Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 2 Year: 2019 Page: 2393-2420
Author(s): Joanna Sniecikowska,Adrian Newman-Tancredi,Marcin Kolaczkowski

Functional Relevance of Biased Signaling at the Angiotensin II Type 1 Receptor

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 11 Issue: 2 Year: 2011 Page: 99-111
Author(s): Douglas G. Tilley

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